L9028-2MG - LK-252
LK-252 | Product ID | L9028 |
| Name | LK-252 |
| Molecular formula | C20H23NO.HCl |
| Description |
a Muscarinic receptors antagonist. Ammonium salt, quinuclidine derivative, , synthetic. |
| Biological activity | pIC50(= -log IC50): M1 (rat brain) = 7.22 M2 (heart) = 6.28 selectivity: [IC50]M2/[IC50]M1 = 8.71 determined by [3H]-QNB binding method, Pirenzepine as standard (unpublished). |
Packaging and Prices
| Packaging | Price (€) | Quantité | Buy Now |
|---|---|---|---|
| 1 x 2mg | 53.00 | ||
| 5 x 2mg | 212.00 | ||
| For quotation of big quantities, please Contact us | |||
Product Technical Documents
 | Safety Data Sheet Available on request, please Contact us Ref. SDS_L9028-2MG : unit price : free of charge |
Chemical and Physical Properties
| Product code | L9028 | Molecular weight | 329.87 Da. |
| Product name | LK-252 | Physical form | |
| CAS No. | 23167-49-9 | Melting point | 173-175 °C. |
| RTECS | Solubility | water. | |
| UNIPROT | Optical Activity | ||
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| PubChem CID | |||
| Purity | min. 98 %. (TLC, NMR). | ||
| Toxicity(LD50) | |||
| Chemical Name | |||
| Storage & Reconstitution Recommandations |
store at +4°C, in dark place. |
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| Savety Recommandations | |||
Bibliographic References
| Product code | L9028 |
| Product name | LK-252 |
- Nilsson et al., J. Med. Chem. (1969). 12:1103-1105
Links
| Product code | L9028 |
| Product name | LK-252 |
| External Links |
PubMed
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Biomedical Citations From PubMed
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Toxicology Citations From PubMed
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