IMPERIALONE | Product ID | L6050 |
| Name | IMPERIALONE |
| Molecular formula | C27H41NO3 |
| Description |
It is a medium-lasting and selective M2 muscarinic receptors antagonist (potency is intermediate between that of L6008 Imperialine and L6032/L6033 chloro-Imperialines). Steroidal Alkaloid , derivative of Imperialine extracted from Petilium eduardi. |
| Biological activity | It presents a M2-selective activity: ED50 on rats under anaesthesia (i.v.) is 0.019 mg/kg (77.5% of Atropine activity). |
Packaging and Prices
| Packaging | Price (€) | Quantité | Buy Now |
|---|---|---|---|
| 1 x 1mg | 125.00 | ||
| 5 x 1mg | 500.00 | ||
| 10 mg | 1 000.00 | ||
| 50 mg | 4 000.00 | ||
| For quotation of big quantities, please Contact us | |||
Product Technical Documents
 | Safety Data Sheet Available on request, please Contact us Ref. SDS_L6050 : unit price : free of charge |
Chemical and Physical Properties
| Product code | L6050 | Molecular weight | 427.61 g/mol |
| Product name | IMPERIALONE | Physical form | Powder |
| CAS No. | 61989-75-1 | Melting point | 228-235 °C |
| RTECS | Solubility | In chloroform Slightly in methanol and ethanol Not well in acetone |
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| UNIPROT | Optical Activity | [alpha]D -31.7° | |
| PubChem SID | |||
| PubChem CID | 90474160 | ||
| Purity | 97% | ||
| Toxicity(LD50) | IVN-MUS LD50: 44 (36-52) mg/kg | ||
| Chemical Name | |||
| Storage & Reconstitution Recommandations |
Store at +4°C, in dark place. |
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| Savety Recommandations | For research use only — not intended for food, diagnostic or therapeutic use |
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Bibliographic References
| Product code | L6050 |
| Product name | IMPERIALONE |
- Nurridinov et al., Chem. Nat. Comp. (1968). 333
- Mirzaev, unbublished results.
Links
| Product code | L6050 |
| Product name | IMPERIALONE |
| External Links |
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