L6258 - IMPERIALINE (3-alpha-Iodo-)
IMPERIALINE (3-alpha-Iodo-) | Product ID | L6258 |
| Name | IMPERIALINE (3-alpha-Iodo-) |
| Molecular formula | C27H42NIO2 |
| Description |
A cardioselective M2-cholinoblocking compound Semi-synthetic alkaloid , derived from base alkaloid Imperialine, isolated from the plant Petilium eduardi and P. raddeanae (Liliaceae fam.) |
| Biological activity | It has M2 cholinoreceptors blocker activity |
Packaging and Prices
| Packaging | Price (€) | Quantité | Buy Now |
|---|---|---|---|
| 20 mg | 148.00 | ||
| 100 mg | 592.00 | ||
| For quotation of big quantities, please Contact us | |||
Product Technical Documents
 | Safety Data Sheet Available on request, please Contact us Ref. SDS_L6258 : unit price : free of charge |
Chemical and Physical Properties
| Product code | L6258 | Molecular weight | 539.53 g/mol |
| Product name | IMPERIALINE (3-alpha-Iodo-) | Physical form | White microcrystalline powder |
| CAS No. | Melting point | 197 - 200 °C | |
| RTECS | Solubility | Easily soluble in chloroform Partly in methanol and acetone |
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| UNIPROT | Optical Activity | Not determined | |
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| Purity | 50% (TLC [silicagel CSC in system: hexan-chloroform-methanol (10:1,5:1), Rf - 0,29]) | ||
| Toxicity(LD50) | IVN-MUS LD50: 51 mg/kg | ||
| Chemical Name | 3alpha-iodo-20beta-oxysevanin-6-one | ||
| Storage & Reconstitution Recommandations |
Reconstitution: soluble in mixture of weak acidic solvent with ethanol while heating (0,1 – 0,3%) soluble in mixture of weak acidic solvent with ethanol.with heating. (0,1 â 0,3%) |
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| Savety Recommandations | For research use only — not intended for food, diagnostic or therapeutic use |
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Bibliographic References
| Product code | L6258 |
| Product name | IMPERIALINE (3-alpha-Iodo-) |
- Roffel A., Meurs H.,Zaagma S., "M-receptors sybtipes: binding, transduction and function", Fundam. Clin. Pharmacol.,1989, Vol. 3., N 4, p.404.
- Mirzaev Yu., Shakirov R. Shakirova U. , "Haloid derivatives of imperialine and its M-cholinoblocking activity", Chim. Prirod. Soedin., 1995, No 2, p. 269 – 271. (Rus.).
Links
| Product code | L6258 |
| Product name | IMPERIALINE (3-alpha-Iodo-) |
| External Links |
PubMed
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Biomedical Citations From PubMed
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Toxicology Citations From PubMed
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